99% Tianeptine sodium letsoai CAS 30123-17-2
Tlhaloso
ITEM | TS'ELISO | RESULT |
Ponahalo | Phofo e tšoeu ho isa ho e mosehla | Phofo e tšoeu ea kristale |
Solubility | Ho qhibiliha ka bolokolohi Metsing le methanol le dichloromethane | E lumellana |
Boitsebiso | Ka IR, Ho tsamaisana le maemo a sebetsang | E lumellana |
(2) E fana ka karabelo ea sodium | E lumellana | |
Litšila A | ≤0.1% | Ha e fumanwe |
Metsoako e amanang | Tšilafalo efe kapa efe e phahameng e le 'ngoe≤0.1% | 0.060% |
Kakaretso ea litšila≤0.4% | 0.36% | |
Residual Solvents (GC) | Acetidin≤ 0.5% | ND |
Dichloromethane≤ 0.06% | ND | |
Methanol≤ 0.3% | ND | |
Acetone≤ 0.5% | 0.29% | |
Acetonitrile≤0.041% | 0.022% | |
Ethanol≤0.5% | ND | |
N, N-dimethylformamide≤0.088% | ND | |
Metsi | ≤ 5.0% | 3.8% |
Assay (HPLC) | 99.0% -101.0% (Ho anhydrousbasis) | 99.70% |
Kopo
Tianeptine sodiumletsoaike tricyclic antidepressant.Mokhoa oa eona oa ho thibela ho tepella maikutlo o fapane le oa li-antidepressants tsa setso tsa tricyclic.E ka eketsa ts'ebetso ea 5-HT ka har'a synaptic cleft.Liphello tsa HT neuronal conduction.Ha ho na kamano bakeng sa li-receptor tsa choline kapa adrenergic.Matla a antidepressant a tšoana le a tricyclics, empa mamello e betere ho feta ea tricyclics.Bakeng sa phekolo ea ho tepella maikutlo ho fokolang, ho leka-lekaneng kapa ho matla haholo, ho tepella maikutlong ha methapo ea pelo le ho itšoara hantle, ho tšoenyeha le ho tepella maikutlong ka 'mele, haholo-holo ho sa phutholoha ha mala, le ho tšoenyeha le ho tepella maikutlong ho bakuli ba nang le joala nakong ea ho tlohela.